Uncovering Kinetic Screen of CCR2 Intracellular Allosteric Antagonists
Kinetic screen of intracellular allosteric antagonists for CCR2 . ‡Ussama I. Choudhry, ‡Tom M. Schubert, ‡Michiel B. Otte, Lisa S. den Hollander* Division of Medicinal Chemistry, Leiden Academic Center for Drug Research, Leiden University, Post Office Box 9502, 2300 RA Leiden, Netherlands INTRODUCTION Chemokines are small molecules with chemoattracting properties[1][2]. These chemokines are … Read more